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PubMed · 10903397

Nonpsychotropic synthetic cannabinoids.

E Pop
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Abstract

Unlike natural cannabinoids which belong to the 6aR - trans series, the synthetic dexanabinol (HU-211), a 6aS-trans enantiomer, does not have affinity toward cannabinoid receptors and is devoid of cannabimimetic activity. On the other hand, dexanabinol demonstrated significant neuroprotective properties which prompted its development as a therapeutic agent. We now present the extension of a series of 6aS-trans cannabinoids with novel derivatives, including water soluble derivatives and congeners of dexanabinol.

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AnimalsCannabinoidsHumansReceptors, CannabinoidReceptors, DrugJournal ArticleReview

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E Pop. 2000. Nonpsychotropic synthetic cannabinoids.. https://doi.org/10.2174/1381612003399446

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