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PubMed · 12666494

[Telithromycin, first ketolide].

Y Van Laethem·J Sternon
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Abstract

Telithromycine is the first ketolide on the market. Its characteristics are the two sites fixation on the bacterial ribosomia and and as a consequence a good activity on the majority of penicillin and macrolides resistant bacteria, included S. pneumonia and S. pyogenes. Telithromycine represents an alternative to beta-lactames and moxifloxacine to treat communautary pneumonia, bacterial pharyngoamygdalitis, suppurative sinusitis and bronchitis. There are nevertheless problems with drugs interactions and risk of resistance development.

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Anti-Bacterial AgentsBacterial InfectionsHumansKetolidesMacrolidesJournal Article

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Y Van Laethem, J Sternon. 2003. [Telithromycin, first ketolide].. https://pubmed.ncbi.nlm.nih.gov/12666494/

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