Methodological implications of simultaneous solid-phase peptide synthesis: a comparison of active esters.

D Hudson

PubMed · 2134048

Methodological implications of simultaneous solid-phase peptide synthesis: a comparison of active esters.

Abstract

Simultaneous competition and comparison methods have been used to compare the activities of a wide variety of reactive esters for solid phase peptide synthesis. The results generally conform to expectations from the literature; the most active being dinitrophenyl esters. Pentafluorophenyl esters provide the most suitable selection for routine use.

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Binding, Competitive Esters Methods Peptides Comparative Study Journal Article

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D Hudson. Methodological implications of simultaneous solid-phase peptide synthesis: a comparison of active esters.. https://pubmed.ncbi.nlm.nih.gov/2134048/

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