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Methodological aspects on drug receptor binding analysis.

A Wahlström
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Abstract

Although drug receptors occur in relatively low concentrations, they can be visualized by the use of appropriate radioindicators. In most cases the procedure is rapid and can reach a high degree of accuracy. Specificity of the interaction is studied by competition analysis. The necessity of using several radioindicators to define a receptor population is emphasized. It may be possible to define isorecptors and drugs with selectivity for one isoreceptor.

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AnimalsHumansProtein BindingRadioligand AssayReceptors, DrugReceptors, OpioidJournal ArticleReview

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BibTeXRIS

A Wahlström. 1978. Methodological aspects on drug receptor binding analysis.. https://doi.org/10.1111/j.1600-0773.1978.tb03223.x

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