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PubMed · 9883617

[Chemotherapeutic agents under study].

S Kawahara
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Abstract

The development of new drugs with strong antituberculous activity and fewer side effects which are not cross-resistant to conventional antituberculosis drugs is urgently desired now. The chemotherapeutic agents under study which are considered a candidate for a new antituberculosis drug are listed below. 1) Rifamycin derivatives: rifabutin, rifapentin, KRM-1648, FCE-22250, 22807, CGP-7040, 27557, 29035, 29861, P-DEA, SPA-S-565, R-76-1. 2) New quinolones: ofloxacin, ciprofloxacin, levofloxacin, sparfloxacin, gatifloxacin, CS-940, Du-6859a. 3) Phenazines: clofazimine, B746, B4101, B4154, B4157. 4) Pyrazinamide derivatives: N-hydroxy pyrazinamide, N-hydroxy pyrazinamide-4-oxide. 5) Nitroimidazole derivatives: metronidazole et al.

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Anti-Infective AgentsAntitubercular AgentsFluoroquinolonesHumansPhenazinesRifamycinsTuberculosisEnglish AbstractJournal ArticleReview

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S Kawahara. 1998. [Chemotherapeutic agents under study].. https://pubmed.ncbi.nlm.nih.gov/9883617/

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