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Soluble polymer-supported convergent parallel library synthesis.

Jung-Mo Ahn·Paul Wentworth·Kim D Janda
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Abstract

Soluble polymer-supported convergent synthesis has for the first time been successfully exploited for parallel library synthesis; sub-libraries of tripeptide iodoarenes and arylboronic acids reacted smoothly in a multipolymer PdII-catalyzed Suzuki coupling reaction to generate a library of bisaryl-linked hexapeptides.

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Combinatorial Chemistry TechniquesOligopeptidesPeptide LibraryPolymersSolubilityJournal ArticleResearch Support, Non-U.S. Gov'tResearch Support, U.S. Gov't, P.H.S.

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Jung-Mo Ahn, Paul Wentworth, Kim D Janda. 2003-02-21. Soluble polymer-supported convergent parallel library synthesis.. https://doi.org/10.1039/b210696e

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