Synthesis of some alkoxybenzamide derivatives as smooth muscle relaxant agents.

S M Rida; F A Ashour; T T Daabees

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PubMed · 31627

Synthesis of some alkoxybenzamide derivatives as smooth muscle relaxant agents.

S M Rida·F A Ashour·T T Daabees

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Abstract

The preparation of 16 new N-substituted p-aminobenzamide derivatives which contain diethylaminoethyl-N-methylpiperazine, piperidine and morpholine moieties were described. Preliminary pharmacological testing of representative compounds showed that some of the prepared compounds possess anticholinergic and antihistaminic activities.

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Animals Benzamides Guinea Pigs Histamine H1 Antagonists In Vitro Techniques Methods Muscle Contraction Muscle Relaxation Muscle, Smooth Parasympatholytics Journal Article

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S M Rida, F A Ashour, T T Daabees. 1978. Synthesis of some alkoxybenzamide derivatives as smooth muscle relaxant agents.. https://pubmed.ncbi.nlm.nih.gov/31627/

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